'Ecstasy' or 3,4-methylene-dioxy-meth-amphetamine (MDMA)
is a psycho-stimulant drug of abuse. Upon consumption, it typically produces
sensations of euphoria, increased sensory awareness, and facilitated social
communication. However, repeated use of MDMA has been strongly linked with
sleep disorders, depressed mood, memory impairment and elevation of anxiety,
impulsiveness and hostility. Since several prescription drugs - chemically
and operationally similar to the "banned" MDMA are considered "safe", the
therapeutic use of MDMA has seemed a coherent idea to some. Further, the
absence of concrete estimates of MDMA doses that are harmful to humans,
and the variability in the nature, intensity and longevity of the impairments
that they cause, have kept the debate on the use of MDMA open.
MDMA operates primarily by affecting the serotonergic
system of the brain, which is known to modulate mood, emotion, sleep and
appetite. In general, high and low levels of the pivotal neuro-transmitter
serotonin have been seen to correspond to positive and negative extremes
of emotion respectively. Under normal conditions of stimulation, the serotonin
released by the serotonin-producing nerve cells triggers responses in the
adjacent neurons. A recycling process called re-uptake then ensues, which
leads to the excess serotonin in the synapse being degraded or reabsorbed.
MDMA alters the serotonin-mechanics by promoting the release and inhibiting
the re-uptake of serotonin. Thus, a short-term serotonin overload results
and causes the characteristic euphoric sensations. Brain-activity in the
human limbic orbito-frontal and antero-temporal structures, which are known
to be involved in emotional processes, has been empirically recorded following
MDMA administration. Thus the spacio-temporal correlation between MDMA
and its immediate emotional effects has sound biochemical and anatomical
backings.
Several experimental studies in animals have shown
that this initial serotonin-overload is followed by a second phase : a
long-lasting decrease in serotonin. This effect could result from a single
large dose or from several moderate doses. It has been seen to last after
abstinence from MDMA, for up to a year in rats and up to 7 years in non-human
primates. Though the exact mechanism of this serotonin-depletion is unknown,
a possible explanation may be obtained from the opponent process theory
of motivation. As an "A-process" (MDMA consumption) lead to an increase
in serotonin levels, a "B-process" was invoked that tried to counter this
effect and maintain homeostasis. With repeated experience (habitual abuse),
this "B-process" increased in magnitude. It thus removed the excess serotonin
more efficiently, ultimately leading to sub-normal serotonin levels. It
is this relatively permanent depletion of serotonin that is the putative
cause of MDMA's long-term neuro-toxicity. Researchers have established
that imbalances in the serotonergic system could cause obsessive compulsive
disorder, sleep onset latency, aggressive behaviors, depression and suicidal
tendencies. It is this chronic and non-ephemeral nature of the pathologies
that has made most scientists take the cautious stand on MDMA usage.
In summary, researchers have elucidated the biochemical
pathways triggered by MDMA, and have also observed a correlation between
the extent of "Ecstasy"-exposure and the severity of cognitive impairment.
Further, histological analyses of brain-tissue from MDMA-administered subjects
have revealed effects like loss of forebrain serotonergic axons and serotonin-system
rewiring. Paradoxically, other amphetamines (Adderall) and chemicals that
target the serotonergic system (Prozac), which could promote this brain-rewiring
equally well, have always been deemed "safe" prescription drugs. Some scientists
suggest that this neuron-rewiring may not be reflective of brain damage
at all. Indeed, an increase of the glial fibrillary acidic protein in the
brain, a reaction diagnostic of chemicals known to damage the brain, has
not been observed for MDMA. In the light of such evidence, it has been
suggested that MDMA administered in controlled doses could possibly alleviate
depression-like syndromes by increasing serotonin levels. Thus, while the
banning of MDMA to discourage its recreational use is justified, claiming
that it causes permanent damage even in small doses is not. The therapeutic
possibilities that MDMA has to offer definitely constitute a promising
area that warrants more research.